Synthesis and SAR of 4-aryl-1-(indazol-5-yl)pyridin-2(1H)ones as MCH-1 antagonists for the treatment of obesity.

Bioorganic & Medicinal Chemistry Letters(2010)

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摘要
The synthesis and SAR of 4-aryl-1-(indazol-5-yl)pyridin-2(1H)ones as MCH-1 antagonists are described.
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关键词
MCH,Obesity,Suzuki,Indazole,Antagonist,Weight loss,SAR
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