N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1)

Bioorganic & Medicinal Chemistry Letters(2008)

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摘要
The synthesis and biological activity of a series of 3-quinolinyl p-aminobenzamide TRPV1 antagonists are reported.
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关键词
TRPV1,Antagonists,Quinolinyl benzamide
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