Discovery Of A New Class Of Non-Imidazole Oxazoline-Based Histamine H-3 Receptor (H3r) Inverse Agonists
CHEMMEDCHEM(2009)
摘要
H(3)R inverse agonists based on an aminopropoxy-phenyloxazoline framework constitute highly valuable druglike lead compounds that display efficacy in a mouse model of recognition memory.
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关键词
cognitive disorders, druglike properties, histamine H-3 receptors, structure-activity relationships, oxazolines
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