Starch nanocapsules containing a novel neutrophil elastase inhibitor with improved pharmaceutical performance.

European Journal of Pharmaceutics and Biopharmaceutics(2018)

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摘要
•ER143-loaded StNC proved as a strategy to improve ER143 pharmaceutical performance.•ER143-loaded StNC showed an improved anti-inflammatory effect.•A QbD approach was successfully applied to obtain ER143-loaded StNC.
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关键词
Starch,Nanocapsules,Neutrophil elastase inhibitors,Topical application
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