Discovery Of Bms-986142: A Reversible Inhibitor Of Bruton'S Tyrosine Kinase (Btk) Conformationally Constrained By Two Locked Atropisomers
Scott Watterson,George De Lucca,Qing Shi,Charles Langevine,Douglas Batt,Qingjie Liu,Myra Beaudoin Bertrand,Hua Gong,Jun Dai,Henry Yip,Peng Li,Dawn Sun,Dauh-Rurng Wu,Chunlei Wang,Yingru Zhang,Sarah Traeger,Mark Pattoli,Stacy Skala,Lihong Cheng,Mary Obermeier, Rodney Vickery,Lorell Discenza, Celia D'Arienzo,Yifan Zhang,Elizabeth Heimrich,Kathleen Gillooly,Tracy Taylor, Claudine Pulicicchio,Kim Mcintyre,Michael Galella,Andrew Tebben,Jodi Muckelbauer,Chiehying Chang,Luisa Salter-Cid,Joel Barrish,Percy Carter,Aberra Fura,James Burke,Joseph Tino ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY(2017)
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