Discovery Of 5 ''-Chloro-N-[(5,6-Dimethoxypyridin-2-Yl)Methyl]-2,2 ':5 ',3 ''-Terpyridine-3 '-Carboxamide (Mk-1064): A Potent, Orally Bioavailable, Selective Orexin 2 Receptor Antagonist That Effectively Promotes Sleep In Preclinical Animal Models
Anthony J. Roecker,Swati P. Mercer,Christopher D. Cox,Mark E. Fraley,John D. Schreier,Justin T. Steen,Pamela L. Tannenbaum,Anthony L. Gotter,Susan L. Garson,Steven V. Fox,C. Meacham Harrell,Joanne Stevens,Wei Lemaire,Joseph G. Bruno,Joyce Stellabott,John D. Higgins,Tamara D. Cabalu,Dan Cui,Thomayant Prueksaritanont,George D. Hartman,Steven D. Young,Christopher J. Winrow,John J. Renger,Paul J. Coleman ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY(2014)
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