Synthetic Procedures from Design and Evaluation of ZD06519, a Novel Camptothecin Payload for Antibody Drug Conjugates

Mark E. Petersen, Michael G. Brant, Manuel Lasalle, Samir Das, Renee Duan, Jodi Wong,Tong Ding, Kaylee J. Wu, Dayananda Siddappa, Chen Fang, Wen Zhang, Alex M. L. Wu, Truman Hirkala-Schaefer,Graham A. E. Garnett,Vincent Fung, Luying Yang, Andrea Hernandez Rojas, Samuel O. Lawn, Stuart D. Barnscher, Jamie R. Rich,Raffaele Colombo

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Synthesis and characterization of free drugs and drug-linkers

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