Imidazopyridines as VLA-4 integrin antagonists
Bioorganic & Medicinal Chemistry Letters(2008)
摘要
The synthesis and SAR of a novel series of imidazopyridine VLA-4 antagonist is described. Compound 15c is a representative example of this series with a human whole blood IC50 of 3nM.
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关键词
VLA-4,Integrin,Imidazopyridine,Phenylalanine
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