Truxillic acid derivatives act as peroxisome proliferator-activated receptor γ activators

Bioorganic & Medicinal Chemistry Letters(2010)

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摘要
Structure-activity relationships of truxillic acid derivatives as subtype-selective PPARγ activators are presented.
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关键词
Nuclear receptors,PPARγ,Truxillic acid derivatives,Reporter gene assay,Molecular docking,Structure–activity relationships
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