Synthesis of quinolinomorphinan-4-ol derivatives as δ opioid receptor agonists.

Yoshihiro Ida,Toru Nemoto,Shigeto Hirayama,Hideaki Fujii,Yumiko Osa,Masayuki Imai,Takashi Nakamura,Toshiyuki Kanemasa,Akira Kato,Hiroshi Nagase

Bioorganic & Medicinal Chemistry（2012）

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摘要

The morphinan derivatives with the 4-hydroxy group (SN-24, 26, 27) showed higher selectivities for the δ receptor over the μ receptor than the corresponding derivatives with the 3-hydroxy group. And they showed high agonist activities for the δ receptor in the [35S]GTPγS binding assay.

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CPM,CBM,c-Pen

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