Design, synthesis and structure-activity relationship of N-substituted tropane muscarinic acetylcholine receptor antagonists.
Bioorganic & Medicinal Chemistry Letters(2012)
摘要
Novel tropane-based, ultra long-acting inhaled muscarinic antagonists: preparation, biological evaluation and developability.
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关键词
Inhaled,Muscarinic antagonist,COPD,Tropane,Quaternary ammonium salts
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