RIP2キナーゼの高強力で選択的阻害剤としての6‐(tert‐ブチルスルホニル)‐N‐(5‐フルオロ‐1H‐インダゾール‐3‐イル)キノリン‐4‐アミン(GSK583)の同定と薬理学的キャラクタリゼーション
A Haile Pamela, J Votta Bartholomew, W Marquis Robert, J Bury Michael, F Mehlmann John, Singhaus Robert, K Charnley Adam, S Lakdawala Ami, A Convery Maire, B Lipshutz David,M Desai Biva, Swift Barbara, A Capriotti Carol, B Berger Scott, K Mahajan Mukesh, A Reilly Michael, J Rivera Elizabeth, H Sun Helen, Nagilla Rakesh, M Beal Allison, N Finger Joshua, N Cook Michael, W King Bryan, T Ouellette Michael, D Totoritis Rachel,Pierdomenico Maria,Negroni Anna,Stronati Laura, Cucchiara Salvatore, Ziolkowski Bartlomiej, Vossenkaemper Anna, T Macdonald Thomas, J Gough Peter,Bertin John, N Casillas Linda Journal of Medicinal Chemistry(2016)
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