Synthesis of Way-163909; a Selective 5-Ht2cr Agonist

SSRN Electronic Journal（2022）

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摘要

A new synthetic approach to derivatives the serotonin 2C receptor (5-HT2CR) agonist WAY-163909 is reported. In addition to the WAY-163909 versions possessing a site that has been shown to accommodate the attachment of linkers without loss of agonist activity are accessible by this approach. An efficient 7 step synthesis with an overall 32% yield is reported.

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关键词

Serotonin,Benzodiazepine,N-heteroannulation,WAY-163909,5-HT2C,5-HT2CR

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