Central Target Engagement and Pharmacodynamic Biomarker Profile for 2 Mg ENX-102, a GABA-A alpha2,3,5 PAM in Development for the Treatment of Generalized Anxiety Disorder

Kimberly Vanover, Pauline Nettesheim, Laura Borghans, Robert-Jan Doll, Estibaliz Arce, Stephen Cunningham, Sean Kipperman, Stephanie Parks, Vikram Sudarsan,Eve Taylor, Philip Kremer,Gabriel Jacobs

NEUROPSYCHOPHARMACOLOGY(2023)

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关键词
Generalized Anxiety Disorder,GABA-A,Positive Allosteric Modulators,Pharmacodynamics
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