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个人简介
The main focus of the current research in the Frølund group is on GHB/CaMK2 pharmacology and the ionotropic GABAA receptors but also covers nACh receptors and the GABA relevant transporters GAT and TauT. The overall goal is to develop molecular probes and novel methodologies to obtain insight into identity, localization, function and therapeutic potential of target receptors/transporters and to match orphan ligands and binding sites with neuroprotection in focus. The approaches comprise structure-activity studies, development of photoligands for determination of localization, mobility and activation of target proteins, and engineered molecular probes for ligand-protein crystallization, identification and probing of binding sites, bioorthogonal chemistry, targeted delivery and rewiring of cell signaling.
研究兴趣
论文共 168 篇作者统计合作学者相似作者
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biorxiv(2024)
Jonas Petersen,Mette Q. Ludwig, Vaida Juozaityte,Pablo Ranea-Robles, Charlotte Svendsen,Eunsang Hwang, Amalie W. Kristensen,Nicole Fadahunsi,Jens Lund, Alberte W. Breum,Cecilie V. Mathiesen, Luisa Sachs,Roger Moreno-Justicia,Rebecca Rohlfs,James C. Ford,Jonathan D. Douros,Brian Finan, Bryan Portillo,Kyle Grose,Jacob E. Petersen,Mette Trauelsen,Annette Feuchtinger,Richard D. DiMarchi,Thue W. Schwartz,Atul S. Deshmukh,Morten B. Thomsen,Kristi A. Kohlmeier,Kevin W. Williams,Tune H. Pers,Bente Frolund,Kristian Stromgaard,Anders B. Klein,Christoffer Clemmensen
Nature (2024)
Communications biologyno. 1 (2023)
Medicinal Chemistry Researchno. 12 (2023): 2587-2587
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作者统计
#Papers: 170
#Citation: 4078
H-Index: 34
G-Index: 57
Sociability: 6
Diversity: 3
Activity: 24
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