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职业迁徙
个人简介
In my research I am interested in elucidating the role of post-translational prenylation of Rab proteins in pathological states, such as cancer and diabetes. As I am chemist, my group works on the synthesis of diverse analogs affecting the Rabs and their prenylating enzyme, Rab geranylgeranyl transferase (GGTase-II). We design the GGTase-II inhibitors and other chemical entities, which allow more in-depth studies of prenylome (e.g. cysteine-targeting moieties, photolabile groups). We are also elaborating new strategies to target particular Rabs, as the inhibition of GGTase-II is too toxic, having an effect on almost all 60 Rabs. We could not do it all ourselves, therefore we are collaborating with colleagues, who generously share their expertise in biology. Our close collaborator from the neighbouring department is Prof. Edyta Gendaszewska-Darmach and her group.
研究兴趣
论文共 49 篇作者统计合作学者相似作者
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Tomasz Sobierajski,Joanna Malolepsza, Marta Pichlak,Edyta Gendaszewska-Darmach,Katarzyna M. Blazewska
DRUG DISCOVERY TODAYno. 7 (2024): 104032-104032
X. H. Liu,J. Lyu,G. Manolikakes,C. E. McKenna, F. Singh,K. Blazewska, X. M. Feng,J. Grimmer, D. Gudat, J. A. Hlina,K. Justyna,B. A. Kashemirov, S. C. Krieg, W. Li
KNOWLEDGE UPDATES 2021/1 (2021)
Knowledge Updates 2021/1 (2021)
KNOWLEDGE UPDATES 2021/1 (2021)
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作者统计
#Papers: 48
#Citation: 963
H-Index: 18
G-Index: 30
Sociability: 5
Diversity: 3
Activity: 15
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